Selected Publications
- The structural diversity of psychedelic drug actions revealed. Ryan H. Gumpper, Manish K. Jain, Kuglae Kim, Renhong Sun, Ning Sun, Zhongli Xu, Jeffrey F. DiBerto, Brian E. Krumm, Nicholas J. Kapolka, H. Ümit Kaniskan, David E. Nichols, Jian Jin, Jonathan F. Fay, Bryan L. Roth. Nature Communications
- Discovery of the first-in-class DOT1L PROTAC degrader. Hyerin Yim, Renhong Sun, Zhongli Xu, Huen Suk Kim, Minjeong Kim, Tao Cao, Ling Xie, Xian Chen, H. Ümit Kaniskan, Jian Jin. European Journal of Medicinal Chemistry
- Discovery of a Potent and Selective Protein Arginine Methyltransferase 5 (PRMT5) PROTAC Degrader. Yue Zhong, Huensuk Kim, Chao Qian, Ling Xie, Xian Chen, Yan Xiong, Jacqueline Hu, Matthew Chen, Ernesto Guccione, Yudao Shen, Jian Jin. Journal of Medicinal Chemistry